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Synthesis and antimalarial activity of cinnamic acid derivatives
(2019)
A peptide coupling reaction between 1-(R)-phenylethylalanine and cinnamic acid derivatives has been
successfully employed for the synthesis of a set of small molecules. The antimalarial activity of these derivative
molecules ...
Synthesis and Antimalarial Activity of 1,4-Disubstituted Piperidine Derivatives
(2020)
In order to prepare, at low cost, new compounds active against Plasmodium falciparum, and
with a less side-effects, we have designed and synthesized a library of 1,4-disubstituted piperidine
derivatives from 4-aminopiperidine ...
Synthesis and evaluation of the antimalarial activity of cinnamic acids derived from piperidine
(2019)
The synthesis and antimalarial activity of 1, 4-aminopiperidine derived cinnamic acids are described. Different
analogs are prepared from reductive amination reactions and SN1 substitutions. These analogs are tested ...